VU Gyvybės mokslų centro autoriaus 'Egidijus Kazlauskas' publikacijų sąrašas

2024
1 Petrauskas, Vytautas; Kazlauskas, Egidijus; Gedgaudas, Marius; Baranauskienė, Lina; Zubrienė, Asta; Matulis, Daumantas. Thermal shift assay for protein–ligand dissociation constant determination // TrAC Trends in Analytical Chemistry. Oxford : Elsevier B.V. ISSN 0165-9936. 2024, vol. 170, art. no. 117417, p. [1-7]. DOI: 10.1016/j.trac.2023.117417. [DB: Science Citation Index Expanded (Web of Science), ScienceDirect]
2 Kairys, Visvaldas; Baranauskienė, Lina; Kazlauskienė, Miglė; Zubrienė, Asta; Petrauskas, Vytautas; Matulis, Daumantas; Kazlauskas, Egidijus. Recent advances in computational and experimental protein-ligand affinity determination techniques // Expert opinion on drug discovery. Abingdon : Taylor and Francis Ltd. ISSN 1746-0441. eISSN 1746-045X. 2024, vol. 19, iss. 6, p. 649-670. DOI: 10.1080/17460441.2024.2349169. [DB: Science Citation Index Expanded (Web of Science), Scopus]
3 Gedgaudas, Marius; Kaziukonytė, Paulina; Kairys, Visvaldas; Mickevičiūtė, Aurelija; Zubrienė, Asta; Brukštus, Algirdas; Matulis, Daumantas; Kazlauskas, Egidijus. Comprehensive analysis of resorcinyl-imidazole Hsp90 inhibitor design // European journal of medicinal chemistry. Issy-les-Moulineaux : Elsevier Masson s.r.l. ISSN 0223-5234. eISSN 1768-3254. 2024, vol. 273, art. no. 116505, p. [1-16]. DOI: 10.1016/j.ejmech.2024.116505. [DB: Science Citation Index Expanded (Web of Science), Scopus]

2023
1 Lingė, Darius; Gedgaudas, Marius; Merkys, Andrius; Petrauskas, Vytautas; Vaitkus, Antanas; Grybauskas, Algirdas; Paketurytė-Latvė, Vaida; Zubrienė, Asta; Zakšauskas, Audrius; Mickevičiūtė, Aurelija; Smirnovienė, Joana; Baranauskienė, Lina; Čapkauskaitė, Edita; Dudutienė, Virginija; Urniežius, Ernestas; Konovalovas, Aleksandras; Kazlauskas, Egidijus; Shubin, Kirill; Schiöth, Helgi B; Chen, Wen-Yih; Ladbury, John E; Gražulis, Saulius; Matulis, Daumantas. PLBD: protein-ligand binding database of thermodynamic and kinetic intrinsic parameters // Database : the journal of biological databases and curation. Oxford : Oxford university press. eISSN 1758-0463. 2023, vol. 2023, art. no. baad040, p. [1-8]. DOI: 10.1093/database/baad040. [DB: Science Citation Index Expanded (Web of Science)]

2022
1 Gedgaudas, Marius; Baronas, Denis; Kazlauskas, Egidijus; Petrauskas, Vytautas; Matulis, Daumantas. Thermott: a comprehensive online tool for protein-ligand binding constant determination // Drug discovery today. Oxford : Elsevier. ISSN 1359-6446. eISSN 1878-5832. 2022, vol. 27, iss. 8, p. 2076-2079. DOI: 10.1016/j.drudis.2022.05.008. [DB: Science Citation Index Expanded (Web of Science), Scopus, Embase, MEDLINE] [IF: 7.400; AIF: 4.500; Q1 (2022 InCities JCR SCIE)]
2 Kaziukonytė, Paulina; Venskūnaitė, Kamilė; Venslauskas, Tomas; Kazlauskas, Egidijus; Gedgaudas, Marius; Žutautė, Ieva; Brukštus, Algirdas. Synthesis and evaluation of Hsp90 inhibition of 1,5-disubstituted imidazoles // 19 Blue Danube symposium on heterocyclic chemistry, August 22-24, 2022, Bratislava, Slovakia : book abstracts. Bratislava, 2022. ISBN 9788082080844. p. 51.

2021
1 Gulla, Aistė; Kazlauskas, Egidijus; Liang, Hong; Strupas, Kęstutis; Petrauskas, Vytautas; Matulis, Daumantas; Eshleman, James R. Heat shock protein 90 inhibitor effects on pancreatic cancer cell cultures // Pancreas. Philadelphia : Lippincot Williams & Wilkins. ISSN 0885-3177. eISSN 1536-4828. 2021, vol. 50, iss. 4, p. 625-632. DOI: 10.1097/MPA.0000000000001807. [DB: Science Citation Index Expanded (Web of Science), Scopus, PubMed] [IF: 3.243; AIF: 7.194; Q3 (2021 InCities JCR SCIE)]
2 Kazlauskas, Egidijus; Petrauskas, Vytautas; Paketurytė, Vaida; Matulis, Daumantas. Standard operating procedure for fluorescent thermal shift assay (FTSA) for determination of protein-ligand binding and protein stability // European biophysics journal. New York : Springer. ISSN 0175-7571. eISSN 1432-1017. 2021, vol. 50, iss. 3-4, p. 373-379. DOI: 10.1007/s00249-021-01537-1. [DB: Science Citation Index Expanded (Web of Science), Scopus, MEDLINE, INSPEC] [IF: 2.095; AIF: 4.632; Q3 (2021 InCities JCR SCIE)]
3 Kaziukonytė, Paulina; Kazlauskas, Egidijus; Brukštus, Algirdas. 4-Isopropyl-6-(1-substituted 1H-imidazol-5-Yl)benzene-1,3-diols as potential Hsp90 inhibitors // Chemistry and chemical technology 2021: 16th international conference of Lithuanian Chemical Society, September 24, 2021, Vilnius : book of abstract. Vilnius. 2021, p. 44. Prieiga per internetą: <http://cct2021.ftmc.lt/wp-content/uploads/2021/09/CCT2021-Book-of-abstracts.pdf>.

2019
1 Kaziukonytė, Paulina; Kazlauskas, Egidijus; Zubrienė, Asta; Brukštus, Algirdas. Synthesis of potential Hsp90 and HDAC multitarget inhibitors // Vilnius University proceedings : Chemistry and chemical technology: Lithuanian chemists conference, 2019 May 16, Lithuanian Academy of Sciences, Vilnius: conference book. Vilnius : Vilniaus universiteto leidykla, 2019. ISBN 9786090701676. p. 75. DOI: 10.15388/CCT.2019.
2 Kairys, Visvaldas; Baranauskienė, Lina; Kazlauskiene, Migle; Matulis, Daumantas; Kazlauskas, Egidijus. Binding affinity in drug design: experimental and computational techniques // Expert opinion on drug discovery. Abingdon : Taylor & Francis. ISSN 1746-0441. eISSN 1746-045X. 2019, vol. 14, iss. 8, p. 755-768. DOI: 10.1080/17460441.2019.1623202. [DB: Current Contents, MEDLINE, Embase, Scopus, Science Citation Index Expanded (Web of Science)] [IF: 4.887; AIF: 3.442; Q1 (2019 InCities JCR SCIE)]

2018
1 Gedgaudas, Marius; Mickevičiūtė, Aurelija; Brukštus, Algirdas; Daunoraitė, Dovilė; Matulis, Daumantas; Kazlauskas, Egidijus. Heat shock protein 90 inhibitors as therapeutic agents against protozoan diseases // Vita Scientia : international conference, 3rd January 2018, Vilnius : conference book. Vilnius : Vita Scientia. ISSN 2538-791X. 2018, p. 32. Prieiga per internetą: <http://www.vitascientia.lt/book> [žiūrėta 2018-04-19].
2 Daunoraitė, Dovilė; Gedgaudas, Marius; Mickevičiūtė, Aurelija; Matulis, Daumantas; Kazlauskas, Egidijus. Cloning, expression and purification of Toxoplasma gondii Hsp90 N domain // Open readings 2018: 61st international conference for students of physics and natural sciences, March 20-23, 2018, Vilnius, Lithuania : programme and abstracts. [S.l.] : [s.n.]. 2018, p. 201. Prieiga per internetą: <http://www.openreadings.eu/wp-content/uploads/2018/03/book.pdf> [žiūrėta 2018-07-19].
3 Synoradzki, Kamil; Miszta, Przemyslaw; Kazlauskas, Egidijus; Mickevičiūtė, Aurelija; Michailovienė, Vilma; Matulis, Daumantas; Filipek, Slawomir; Bieganowski, Pawel. Interaction of the middle domains stabilizes Hsp90α dimer in a closed conformation with high affinity for p23 // Biological chemistry. Berlin : Walter de Gruyter GmbH. ISSN 1431-6730. eISSN 1437-4315. 2018, vol. 399, no 4, p. 337-345. DOI: 10.1515/hsz-2017-0172. [DB: Scopus, Science Citation Index Expanded (Web of Science)] [IF: 3.014; AIF: 4.417; Q2 (2018 InCities JCR SCIE)]

2015
1 Dudutienė, Virginija; Matulienė, Jurgita; Smirnov, Alexey; Timm, David Daniel; Zubrienė, Asta; Baranauskienė, Lina; Morkūnaitė, Vaida; Smirnovienė, Joana; Michailovienė, Vilma; Juozapaitienė, Vaida; Mickevičiūtė, Aurelija; Kazokaitė, Justina; Bakšytė, Sandra; Kasiliauskaitė, Aistė; Jachno, Jelena; Revuckienė, Jurgita; Kišonaitė, Miglė; Pilipuitytė, Vilma; Ivanauskaitė, Eglė; Milinavičiūtė, Goda; Smirnovas, Vytautas; Petrikaitė, Vilma; Kairys, Visvaldas; Petrauskas, Vytautas; Norvaišas, Povilas; Lingė, Darius; Gibieža, Paulius; Čapkauskaitė, Edita; Zakšauskas, Audrius; Kazlauskas, Egidijus; Manakova, Elena; Gražulis, Saulius; Ladbury, J. E.; Matulis, Daumantas. Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX // Chemistry and chemical technology 2015 : international conference of Lithuanian Chemical Society, dedicated to Professor Vitas Daukšas on his 80th birth anniversary, Vilnius, Lithuania, January 23, 2015 : programme and proceedings of the international conference. Vilnius : Vilnius University, 2015. ISBN 9786094594618. p. 25.

2014
1 Brukštus, Algirdas; Kazlauskas, Egidijus; Petrikas, Herkus; Petrikaitė, Vilma; Čikotienė, Inga; Matulis, Daumantas. Synthesis and biological evaluation of 6-(5-aryl-1,2,3-thiadiazol-4-yl)-4-isopropylbenzene-1,3-dioles as inhibitors of HSP90 chaperone // Chemistry and chemical technology : proceedings of the international conference, Kaunas, 25 April 2014. Kaunas : Technologija. ISSN 2351-5643. 2014, p. 210-211.
2 Dudutienė, Virginija; Matulienė, Jurgita; Smirnov, Alexey; Timm, David Daniel; Zubrienė, Asta; Baranauskienė, Lina; Morkūnaitė, Vaida; Smirnovienė, Joana; Michailovienė, Vilma; Juozapaitienė, Vaida; Mickevičiūtė, Aurelija; Kazokaitė, Justina; Bakšytė, Sandra; Kasiliauskaitė, Aistė; Jachno, Jelena; Revuckienė, Jurgita; Kišonaitė, Miglė; Pilipuitytė, Vilma; Ivanauskaitė, Eglė; Milinavičiūtė, Goda; Smirnovas, Vytautas; Petrikaitė, Vilma; Kairys, Visvaldas; Petrauskas, Vytautas; Norvaišas, Povilas; Lingė, Darius; Gibieža, Paulius; Čapkauskaitė, Edita; Zakšauskas, Audrius; Kazlauskas, Egidijus; Manakova, Elena; Gražulis, Saulius; Ladbury, John E.; Matulis, Daumantas. Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX // Journal of medicinal chemistry. Washington : American Chemical Society. ISSN 0022-2623. eISSN 1520-4804. 2014, vol. 57, no 22, p. 9435-9446. DOI: 10.1021/jm501003k. [DB: Science Citation Index Expanded (Web of Science), CABI Abstracts Databases, Chimica, Scopus, MEDLINE, Embase] [IF: 5.447; AIF: 2.621; Q1 (2014 InCities JCR SCIE)]

2013
1 Zubrienė, Asta; Gylytė, Joana; Morkūnaitė, Vaida; Kazlauskas, Egidijus; Baranauskienė, Lina; Čapkauskaitė, Edita; Dudutienė, Virginija; Jogaitė, Vaida; Michailovienė, Vilma; Kazokaitė, Justina; Timm, David Daniel; Petrauskas, Vytautas; Matulienė, Jurgita; Matulis, Daumantas. Thermodynamics of anticancer drug lead binding to target proteins by thermal shift assay // European biophysics journal with biophysics letters: 9th EBSA European Biophysics Congress, 13-17 July 2013, Lisbon, Portugal - abstracts. New York : Springer. ISSN 0175-7571. eISSN 1432-1017. 2013, vol. 42, suppl. 1, art. no. P-303, p. S114. DOI: 10.1007/s00249-013-0917-x. [DB: Science Citation Index Expanded (Web of Science)] [IF: 2.474; AIF: 3.289; Q3 (2013 InCities JCR SCIE)]
2 Petrikaitė, Vilma; Kazlauskas, Egidijus; Matulis, Daumantas. Thermodynamics of Aryl-dihydroxyphenyl-thiadiazole inhibitor series binding to molecular chaperone Hsp90 // Epigenetics – Bench to Bedside. COST Action TD0905 : Program and Abstract Book : October 30-31, 2013, Vilnius, Lithuania / Organizers: Daumantas Matulis, Jurgita Revuckienė ; Institute of Biotechnology. Vilnius University. Biothermodynamics & Drug Design Dept. European Cooperation in Science and Technology. Vilnius : Institute of Biotechnology. Vilnius University. 2013, p. 32, no. ps8.
3 Kazlauskas, Egidijus; Petrikaitė, Vilma; Matulis, Daumantas. Thermodynamics of Aryl-dihydroxyphenyl-thiadiazole Inhibitor Series Binding to Molecular Chaperone Hsp90 // CEEC-TAC2 – 2nd Central and Eastern European Conference on Thermal Analysis and Calorimetry : Book of Abstracts : 27-30 August 2013, Vilnius, Lithuania / Editors: Andrei Rotaru, Daumantas Matulis. [S. l.] : Central and Eastern European Committee for Thermal Analysis and Calorimetry, 2013. ISBN 978-3-940237-33-0. p. 376, no. ps3.30.

2012
1 Matulis, Daumantas (autorius, išradimo); Čikotienė, Inga (autorius, išradimo); Kazlauskas, Egidijus (autorius, išradimo); Matulienė, Jurgita (autorius, išradimo). 5-aryl-4-(5-substituted 2,4-dihydroxyphenyl)-1,2,3-thiadiazoles as inhibitors of HSP90 chaperone and the intermediates for production thereof. EP2268626 B1. Prieiga per internetą: <http://www.freepatentsonline.com/EP2268626.pdf> [žiūrėta 2012-05-02].
2 Giessrigl, Benedikt; Krieger, Sigurd; Rosner, Margit; Huttary, Nicole; Saiko, Phillipp; Alami, Mouad; Messaoudi, Samir; Peyrat, Jean-Francois; Maciuk, Alexandre; Gollinger, Michaela; Kopf, Sabine; Kazlauskas, Egidijus; Mazal, Peter; Szekeres, Thomas; Hengstschläger, Markus; Matulis, Daumantas; Jäger, Walter; Krupitza, Georg. Hsp90 stabilizes Cdc25A and counteracts heat shock-mediated Cdc25A degradation and cell-cycle attenuation in pancreatic carcinoma cells // Human molecular genetics. Oxford : Oxford University Press. ISSN 0964-6906. 2012, Vol. 21, no. 21, p. 4615-4627. DOI: 10.1093/hmg/dds303. [DB: Science Citation Index Expanded (Web of Science), BIOSIS Previews, Biological Abstracts] [IF: 7.692; AIF: 4.379; Q1 (2012 InCities JCR SCIE)]
3 Matulis, Daumantas (autorius, išradimo); Čikotienė, Inga (autorius, išradimo); Kazlauskas, Egidijus (autorius, išradimo); Matulienė, Jurgita (autorius, išradimo). 5-aryl-4-(5-substituted 2,4-dihydroxyphenyl)-1,2,3-thiadiazoles as inhibitors of Hsp90 chaperone and the intermediates for production thereof : patent no.: US 8,314,132 B2 / inventors: Matulis; Daumantas (Vilnius, LT), Cikotiene; Inga (Vilnius, LT), Kazlauskas; Egidijus (Vilnius, LT), Matuliene; Jurgita (Vilnius, LT). Appl. no.: 12/990,551. 2012-11-20.
4 Sharp, Swee Y.; Roe, S. Mark; Kazlauskas, Egidijus; Čikotienė, Inga; Workman, Paul; Matulis, Daumantas; Prodromou, Chrisostomos. Co-Crystalization and In Vitro Biological Characterization of 5-Aryl-4-(5-Substituted-2-4-Dihydroxyphenyl)-1,2,3-Thiadiazole Hsp90 Inhibitors // PLoS ONE [Elektroninis išteklius]. San Francisko : Public Library of Science. ISSN 1932-6203. 2012, Vol. 7, iss. 9, Art. No. e44642. DOI: 10.1371/journal.pone.0044642. [DB: Science Citation Index Expanded (Web of Science), PubMed, MEDLINE, Scopus, AGRICOLA, PyscINFO, Zoological Record, Embase] [IF: 3.730; AIF: 6.803; Q1 (2012 InCities JCR SCIE)]
5 Kazlauskas, Egidijus; Petrikaitė, Vilma; Michailovienė, Vilma; Revuckienė, Jurgita; Matulienė, Jurgita; Grinius, Leonas; Matulis, Daumantas. Thermodynamics of Aryl-Dihydroxyphenyl-Thiadiazole Binding to Human Hsp90 // PLoS One. San Francisco : Public Library of Science. ISSN 1932-6203. 2012, vol. 7, no. 5, Art. No. e36899 (12 p.). DOI: 10.1371/journal.pone.0036899. [DB: DOAJ, GeoRef, Food Science & Technology Abstracts (IFIS), Zoological Record, PyscINFO, AGRICOLA, Scopus, MEDLINE, Science Citation Index Expanded (Web of Science)] [IF: 3.730; AIF: 6.803; Q1 (2012 InCities JCR SCIE)]

2011
1 Zubrienė, Asta; Kazlauskas, Egidijus; Michailovienė, Vilma; Matulis, Daumantas. Towards intrinsic binding thermodynamics // European biophysics journal with biophysics letters: 8th EBSA European Biophysics Congress, August 23rd–27th 2011, Budapest, Hungary : abstracts. New York : Springer. ISSN 0175-7571. 2011, vol. 40, suppl. 1, art. no. P-110, p. 66. DOI: 10.1007/s00249-011-0734-z. [DB: Science Citation Index Expanded (Web of Science)] [IF: 2.139; AIF: 3.403; Q3 (2011 InCities JCR SCIE)]
2 Zubrienė, Asta; Kazlauskas, Egidijus; Baranauskienė, Lina; Petrauskas, Vytautas; Matulis, Daumantas. Isothermal titration calorimetry and thermal shift assay in drug design // European pharmaceutical review. Brasted, Kent : Russell Publishing Ltd. ISSN 1360-8606. 2011, Vol. 16, iss. 3, p. 56-59. Prieiga per internetą: <https://www.europeanpharmaceuticalreview.com/article/7622/isothermal-titration-calorimetry-and-thermal-shift-assay-in-drug-design/> [žiūrėta 2017-09-25]. [DB: Embase, Scopus]